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1Main
2
3TAK-242 (resatorvid)Sepsis1TLR4
4SNT-MC17 (idebenone)Friedreich's AtaxiaSantheraIII
5AMG706 (motesanib)CancerAMGNKinaseIII
6TAK-379 failure
7TAK-013EndometriosisLHRH antagonist
8Omontys (fka Hematide, peginesatide)AnemiaAffymxaEPO
9Zafatek (fka SYR-472) (trelagliptin)Type 2 Diabetes100% (Furiex acquisition)DPP4Approved in Japan
10Mepact (mifamurtide)Osteosarcoma1EU 09
11Basen (voglibose)Type 2 Diabetes1
12Edarbi (TAK-491 (azilsartan)) TAK-536?Hypertension1ARBNDA USNCE
13ferumoxytolAnemiaAMAG; deal terminatedJapan rights only
14Lotriga (TAK-085)HypertriglyceridemiaPronovaEPA/DHA
15GalantamineAlzheimer'sJNJ
16
17TAK-583Neuropathic Paindiscontinued in 2008
18ATL-692 (cetilistat)ObesityNorginelipase inhibitorIII JP
19MCC-135 (caldaret)CHFCa++ uptake enhancer
20TAK-370 (mosapride)GERD5-HT4 agonistapproved in some Asian countries?
21IY-81149PPI
22TAK-428Diabetic neuropathy1oral NGF agonistII US/EU
23TAK-442 (letaxaban)Thromboembolism1Factor XaII US/EU
24TAK-654 (sipoglitazar)Type 2 DiabetesPPAR
25TAK-700 (orteronel)HRPC1Androgen inhibitorII
26MLN0518 (tandutinib)Glioblastoma1FLT3II
27Lu AA24530 (tedatioxetine)DepressionLUN DCII
28MLN8237 (alisertib)NHL1AuroraII
29CBP501NSCLCCanBascalmodulinII
30AMG665 (conatumumab)CancerAMGNDR5I
31AMG386 (trebananib)CancerAMGNAngiopoietinI
32AMG479 (ganitumab)CancerAMGNIGF-1RI
33TAK-100Type 2 Diabetes1DPP4I
34TAK-591Hypertension1ARBI
35TAK-329Glucokinase1I
36TAK-875Type 2 Diabetes1GPR40II
37TAK-851HPV1II US/EUTopical
38TAK-683 (metastin)HRPC1KISS1R agonistI
39TAK-448 (metastin)HRPC1KISS1RI
40TAK-285Cancer1HER2I
41TAK-802Hypoactive bladderacetylcholinesterase