ABCDEFGH
1Main
2BrandGenericIndicationApprovedEconomicsMOA
3TamifluoseltamivirInfluenza1999GileadNeuraminidase
4ValcytevalganciclovirHerpes3/9/2001
5
6Dalcetrapib fails.
7July 2013: aleglitazar stopped
82014: bitopertin (RG1678) fails.
9
10
11
127166, triple reuptake inhibitor for depression, abandoned.
137351, TAAR1 partial agonist for depression, abandoned
14R1579 (carmegliptin)T2DII1DPP-IVNCE
15R667 (palovarotene)EmphysemaII1Nuclear Receptor AgonistNCE
16RG3487Alzheimer's, SchizophreniaII1Alpha-7NCE
17RG3484Cervical NeoplasiaII1HPV16 vaccineVaccine
18R7128HCVIIVRUSNucleoside PolymeraseANDS, VX-222NCE
19R7227HCVIITMNProtease Inhibitor11/09: Safety issueNCE
20R7234T2DI111-beta-HSDNCE
21R4929T2DI111-beta-HSDNCE
22R7089T2DI1Y2R peptide agonistNCE
23RG7426T1DI1NCE
24RO4998452T2DII1NCE
25EVT101Treatment Resistant DepressionII1NMDA?NCE?
26RG7090 (basimglurant)DepressionII1mGluR5Outlicensed to Noema PharmaNCE
27R7201 (tofogliflozin)T2DIIChugaiSGLT2NCE
28RG7423Solid TumorsII1Small MoleculeNCE
29R3637 (lebrikizumab)AsthmaIILLYAnti IL-13Antibody
30RG3638 (onartuzumab)Solid TumorsIII1MetMabAntibody
31RG3639 (dulanermin)Solid TumorsIIAMGNDR5?Protein
32R7376 (PLX5568)Polycystic Kidney DiseaseIIPlexxiconRAF kinase inhibitorNCE
33R1512PVDIGenmabSelectinAntibody
34ABT-263 (navitoclax) RG7601?R/R CLLIIABTBcl-2NCE
35R7417 (lampalizumab)AMDI1Anti-Factor-DNCE
36R7273DyslipidemiaI1ABCA1 inducerNCE