|
Main | | | | | | | |
| Brand | Generic | Indication | Approved | Economics | MOA | |
| Tamiflu | oseltamivir | Influenza | 1999 | Gilead | Neuraminidase | |
| Valcyte | valganciclovir | Herpes | 3/9/2001 | | | |
| | | | | | | |
| Dalcetrapib fails. | | | | | | |
| July 2013: aleglitazar stopped | | | | | | |
| 2014: bitopertin (RG1678) fails. | | | | | | |
| | | | | | | |
| | | | | | | |
| | | | | | | |
| 7166, triple reuptake inhibitor for depression, abandoned. | | | | | | |
| 7351, TAAR1 partial agonist for depression, abandoned | | | | | | |
| R1579 (carmegliptin) | T2D | II | 1 | DPP-IV | | NCE |
| R667 (palovarotene) | Emphysema | II | 1 | Nuclear Receptor Agonist | | NCE |
| RG3487 | Alzheimer's, Schizophrenia | II | 1 | Alpha-7 | | NCE |
| RG3484 | Cervical Neoplasia | II | 1 | HPV16 vaccine | | Vaccine |
| R7128 | HCV | II | VRUS | Nucleoside Polymerase | ANDS, VX-222 | NCE |
| R7227 | HCV | I | ITMN | Protease Inhibitor | 11/09: Safety issue | NCE |
| R7234 | T2D | I | 1 | 11-beta-HSD | | NCE |
| R4929 | T2D | I | 1 | 11-beta-HSD | | NCE |
| R7089 | T2D | I | 1 | Y2R peptide agonist | | NCE |
| RG7426 | T1D | I | 1 | | | NCE |
| RO4998452 | T2D | II | 1 | | | NCE |
| EVT101 | Treatment Resistant Depression | II | 1 | NMDA? | | NCE? |
| RG7090 (basimglurant) | Depression | II | 1 | mGluR5 | Outlicensed to Noema Pharma | NCE |
| R7201 (tofogliflozin) | T2D | II | Chugai | SGLT2 | NCE | |
| RG7423 | Solid Tumors | II | 1 | Small Molecule | NCE | |
| R3637 (lebrikizumab) | Asthma | II | LLY | Anti IL-13 | Antibody | |
| RG3638 (onartuzumab) | Solid Tumors | III | 1 | MetMab | Antibody | |
| RG3639 (dulanermin) | Solid Tumors | II | AMGN | DR5? | Protein | |
| R7376 (PLX5568) | Polycystic Kidney Disease | II | Plexxicon | RAF kinase inhibitor | NCE | |
| R1512 | PVD | I | Genmab | Selectin | Antibody | |
| ABT-263 (navitoclax) RG7601? | R/R CLL | II | ABT | Bcl-2 | NCE | |
| R7417 (lampalizumab) | AMD | I | 1 | Anti-Factor-D | NCE | |
| R7273 | Dyslipidemia | I | 1 | ABCA1 inducer | NCE | |