| A | B | C | D | E | F | G | H | I | |
|---|---|---|---|---|---|---|---|---|---|
| 1 | Main | ||||||||
| 2 | Brand | Generic | Indication | MOA | Phase | Active? | Company | Notes | |
| 3 | SEP-363856 | ulotaront | Schizophrenia | TAAR agonist | III | YES | 4506 JP | Phase II n=245, 50mg, 75mg or PBO. -17.2 points vs -9.7 points at 4 weeks. | |
| 4 | SAGE | ||||||||
| 5 | tedatioxetine | TAK/LUN | |||||||
| 6 | TAK-041/NBI-846 | Depression | GPR139 agonist | II | YES | ||||
| 7 | TAK-653/NBI-845 | Depression | AMPA agonist | ||||||
| 8 | amantadine | ||||||||
| 9 | MK-1942 | TRD | YES | MRK | |||||
| 10 | CVL-231 | emraclidine | Schizophrenia | M4 PAM | II | YES | CERE | ||
| 11 | NBI-1117568 | Schizophrenia | M4 PAM | II | YES | NBIX | |||
| 12 | MK-8189 | Schizophrenia | PDE10A inhibitor | II | YES | MRK | |||
| 13 | RP5063 | brilaroxazine | Schizophrenia | D2 partial agonist | III | YES | Reviva Pharmaceuticals | ||
| 14 | KarXT | xanomeline, trospium | Schizophrenia | M4 PAM | III | YES | KRTX | ||
| 15 | CPL500036 | Schizophrenia | PDE10A inhibitor | II | YES | Celon Pharma SA | |||
| 16 | Falkieri | esketamine | Bipolar Depression | NMDA | YES | Celon Pharma SA | |||
| 17 | BI 425809 | Schizophrenia | GlyT1 inhibitor | II | YES | Boehringer Ingelheim | |||
| 18 | TV-44749 | olanzapine | Schizophrenia | D2 antagonist | III | YES | TEVA | ||
| 19 | TPN672 | Schizophrenia | D2 antagonist | I | YES | Jiangsu Kanion | |||
| 20 | agomelatine | ||||||||
| 21 | TAK-831/NBI-1065844 | luvadaxistat | CIS Schizophrenia | DAAO inhibitor | TAK/NBIX | ||||
| 22 | RL-007 | CIS Schizophrenia | GABA/nicotinic | I | YES | Recognify | |||
| 23 | HS-10380 | Jiangsu Hansoh | |||||||
| 24 | LYN-005 | risperidone | Schizophrenia | D2 antagonist | I | YES | Lyndra Therapeutics | ||
| 25 | JX11502MA | Schizophrenia | Zhejiang Jingxin | ||||||
| 26 | LY03010 | paliperidone palmitate | Schizophrenia | ||||||
| 27 | vabicaserin | ||||||||
| 28 | PF-02545920 | ||||||||
| 29 | RG1678 | ||||||||
| 30 | MK-0249 | ||||||||
| 31 | encenicline | ||||||||
| 32 | LY404039 | ||||||||
| 33 | CX516 | ||||||||
| 34 | SR48692 | ||||||||
| 35 | SR142801 | ||||||||
| 36 | SR141716 | ||||||||
| 37 | L-745870 | ||||||||
| 38 | SCH39166 | ||||||||
| 39 | M100907 | ||||||||
| 40 | TAK-063 |