ABC
1
2Brand NameINCB7839
3Generic Name
4IndicationSolid Tumors, Breast Cancer
5MechanismSheddase Inhibitor; synergy with herceptin given the ability to maintain HER2 on cells by inhibiting sheddase activity (which may make them more susceptible to Herceptin)
6AdministrationMTD unknown
7Competition
8Economics
9IP
10History
11Clinical Trials
12Phase Ib / IIa solid tumors
13maximal tolerated dose has yet to be reached
14
15Phase Ib / IIa Breast Cancer
16plan initiation